Product Name: Carfilzomib (PR-171)
Subtitle: Proteasome inhibitor,epoxomicin analog
Biological Activity: Biological Activity of Carfilzomib (PR-171)Description Carfilzomib (PR-171) is an irreversible inhibitor of proteasome with IC50 of <5 nM. Targets Proteasome IC50 5 nM
SMLES: CC(C)C[C@@H](C(=O)[C@]1(CO1)C)NC(=O)[C@H](CC2=CC=CC=C2)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC3=CC=CC=C3)NC(=O)CN4CCOCC4
CAS NO: 1009298-09-2
Standard In CHIKey: sFRP-1 inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C40H57N5O7
M.Wt: 719.91
General Tips: for obtaining a higher concentration: Please warm the tube at 37 °C for 10 minutes and/or shake it in the ultrasonic bath for a while.Stock solution can be stored below -20°C for several months.PubMed ID:http://jpet.aspetjournals.org/content/259/3/1379
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: Carfilzomib