Product Name: PF 429242
Subtitle:
Biological Activity: Biological Activity of PF 429242Reversible, competitive inhibitor of sterol regulatory element-binding protein (SREBP) site 1 protease (IC50 = 0.175 μM). Selective for site 1 protease against a panel of serine proteases. Inhibits rate of cholesterol
SMLES: N/A
CAS NO: 700878-19-9
Standard In CHIKey: TAK1 inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C25H35N3O2.2HCl
M.Wt: 482.49
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/271/3/1299
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 50 mM in water and to 50 mM in DMSO
Storage: Desiccate at RT
Purity: >98%
Chemical Name: 4-[(Diethylamino)methyl]-N-[2-(2-methoxyphenyl)ethyl]-N-(3R)-3-pyrrolidinylbenzamide