Product Name: 1-Azakenpaullone
Subtitle: GSK-3β inhibitor,potent and selective,cell-permeable
Biological Activity: Biological Activity of 1-AzakenpaulloneDescription 1-Azakenpaullone is a potent and selective inhibitor of GSK-3β with IC50 of 18 nM. Targets GSK-3β IC50 18 nM
SMLES: C1C2=C(C3=C(C=CC=N3)NC1=O)NC4=C2C=C(C=C4)Br
CAS NO: 816432-15-2
Standard In CHIKey: IRAK inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C15H10BrN3O
M.Wt: 328.16
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/271/1/353
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: (1S,3R,4R,5R)-1,3-bis[[(E)-3-(3,4-dihydroxyphenyl)prop-2-enoyl]oxy]-4,5-dihydroxycyclohexane-1-carboxylic acid