Product Name: 8-CPT-2Me-cAMP, sodium salt
Subtitle: EPAC agonist, selective
Biological Activity: Biological Activity of 8-CPT-2Me-cAMP, sodium saltSelective activator of Epac, the cAMP-sensitive guanine nucleotide-exchange factor for Rap1 and Rap2. Activates Epac1 (EC50 = 2.2 μM), but not PKA (EC50 > 10 μM). Stimulates Epac-mediated Ca2+
SMLES:
CAS NO: 180977-34-8
Standard In CHIKey: mTOR inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C17H16ClN5O6PS.Na
M.Wt: 507.82
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/273/3/1307
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in water
Storage: Desiccate at -20℃
Purity: >98%
Chemical Name: 8-(4-Chlorophenylthio)-2-O-methyladenosine-3,5-cyclic monophosphate sodium salt