Product Name: A 784168
Subtitle: TRPV1 antagonist,potent and selective
Biological Activity: Biological Activity of A 784168Potent TRPV1 antagonist (IC50 = 25 nM for inhibition of TRPV1 activation by 50 nM capsaicin). Displays no activity against a range of receptors, including TRPA1, GABA, opioid, and purinergic receptors.
SMLES:
CAS NO: 1538604-68-0
Standard In CHIKey: p97 inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C19H15F6N3O3S
M.Wt: 479.4
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/272/2/901
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in DMSO and to 50 mM in ethanol
Storage: Store at RT
Purity: >98%
Chemical Name: 3,6-Dihydro-3-(trifluoromethyl)-N-[4-[(trifluoromethyl)sulfonyl]phenyl]-[1(2H),2-bipyridine]-4-carboxamide