Product Name: A 841720
Subtitle: mGluR1 antagonist, non-competitive
Biological Activity: Biological Activity of A 841720Potent, non-competitive mGlu1 receptor antagonist that displays 34-fold selectivity over mGlu5 (IC50 values are 10 and 342 nM respectively). Displays no significant activity at a range of other GPCRs, ion channels and transp
SMLES:
CAS NO: 1156-19-0
Standard In CHIKey: DNA-PK inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C17H21N5OS
M.Wt: 343.45
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/270/3/1086
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 50 mM in DMSO and to 50 mM in ethanol
Storage: Store at RT
Purity: >98%
Chemical Name: 9-(Dimethylamino)-3-(hexahydro-1H-azepin-1-yl)pyrido[3,2:4,5]thieno[3,2-d]pyrimidin-4(3H)-one