Product Name: BL 1249
Subtitle: Putative activator of potassium TREK-1
Biological Activity: Biological Activity of BL 1249Putative potassium channel activator; thought to act as a K2P2.1 (TREK-1) channel opener. Exhibits selectivity for bladder over vascular tissue in vitro and in vivo (EC50 values are 1.26 and 21.0 μM for cultured bladder
SMLES:
CAS NO: 21416-43-3
Standard In CHIKey: LRRK2 inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C17H17N5
M.Wt: 291.35
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/274/2/735
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in 1eq. NaOH and to 100 mM in DMSO
Storage: Store at -20℃
Purity: >98%
Chemical Name: 5,6,7,8-Tetrahydro-N-[2-(2H-tetrazol-5-yl)phenyl]-1-naphthalenamine