Product Name: CEP-18770
Subtitle: Proteasome inhibitor
Biological Activity: Biological Activity of CEP-18770Description CEP-18770 is a novel orally-active inhibitor of the chymotrypsin-like activity of the proteasome with a cellular IC50 value of 3.8 nM. Targets proteasome IC50 3.8 nM
SMLES: B(C(CC(C)C)NC(=O)C(C(C)O)NC(=O)C1=CC=CC(=N1)C2=CC=CC=C2)(O)O
CAS NO: 885060-09-3
Standard In CHIKey: Aromatase inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C21H28BN3O5
M.Wt: 413.3
General Tips: for obtaining a higher concentration: Please warm the tube at 37 °C for 10 minutes and/or shake it in the ultrasonic bath for a while.Stock solution can be stored below -20°C for several months.PubMed ID:http://jpet.aspetjournals.org/content/26/1/1
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: [(1R)-1-[[(2S,3R)-3-hydroxy-2-[(6-phenylpyridine-2-carbonyl)amino]butanoyl]amino]-3-methylbutyl]boronic acid