Product Name: CI 966 hydrochloride
Subtitle:
Biological Activity: Biological Activity of CI 966 hydrochlorideSelective inhibitor of the GABA transporter GAT-1 (IC50 values are 0.26 and 1.2 μM at cloned human and rat GAT-1 respectively). Displays over 200-fold selectivity over GAT-2 and GAT-3. Centrally active upon sy
SMLES: FC(F)(C1=CC=C(C=C1)C(C2=CC=C(C(F)(F)F)C=C2)OCCN3CCC=C(C(O)=O)C3)F.Cl
CAS NO: 153777-70-9
Standard In CHIKey: NUQWSOWKRTZJTO-UHFFFAOYSA-NNeprilysin inhibitors
Standard InChI: InChI=1S/C23H21F6NO3.ClH/c24-22(25,26)18-7-3-15(4-8-18)20(16-5-9-19(10-6-16)23(27,28)29)33-13-12-30-11-1-2-17(14-30)21(31)32;/h2-10,20H,1,11-14H2,(H,31,32);1H
Typrof Compound:
Appearance:
Formula: C23H21F6NO3.HCl
M.Wt: 509.87
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/273/2/967
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 10 mM in ethanol and to 100 mM in DMSO
Storage: Desiccate at RT
Purity: >98%
Chemical Name: 1-[2-[bis[4-(Trifluoromethyl)phenyl]methoxy]ethyl]-1,2,5,6-tetrahydropyridine-3-carboxylic acid hydrochloride