Product Name: Clobenpropit dihydrobromide
Subtitle:
Biological Activity: Biological Activity of Clobenpropit dihydrobromideAn extremely potent histamine H3 antagonist/inverse agonist (pA2=9.93). Also displays partial agonist activity at H4 receptors; induces eosinophil shape change with an EC50 of 3 nM. Also available as part
SMLES: ClC1=CC=C(C=C1)C/N=C(N)SCCCC2=CN=CN2.Br.Br
CAS NO: 17575-22-3
Standard In CHIKey: PERK inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C14H17ClN4S.2HBr
M.Wt: 470.65
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/27/2/125
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in water
Storage: Store at RT
Purity: >98%
Chemical Name: N-(4-Chlorobenzyl)-S-[3-(4(5)-imidazolyl)propyl]isothiourea dihydrobromide