Product Name: JNJ 5207787
Subtitle:
Biological Activity: Biological Activity of JNJ 5207787Selective NPY Y2 antagonist (IC50 = 0.1 μM). Displays 100-fold selectivity over NPY Y1, Y4 and Y5 receptors; also displays selectivity against a panel of 50 receptors, ion channels and transporters. Brain penetrant.
SMLES: O=C(/C=CC1=CC=CC(C#N)=C1)N(C2=CC=C3C(N(C(C)=O)CC3)=C2)C4CCN(CC4)CCC5CCCC5
CAS NO: 97657-92-6
Standard In CHIKey: HIV inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C32H38N4O2
M.Wt: 510.67
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/264/1/397
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 10 mM in DMSO with gentle warming and to 10 mM in ethanol with gentle warming
Storage: Store at RT
Purity: >98%
Chemical Name: (2E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-3-(3-cyanophenyl)-N-[1-(2-cyclopentylethyl)-4-piperidinyl]-2-propenamide