Product Name: Kenpaullone
Subtitle:
Biological Activity: Biological Activity of KenpaullonePotent inhibitor of CDK1/cyclin B and GSK-3β (IC50 values are 0.4 and 0.23 μM respectively). Also inhibits CDK2/cyclin A, CDK2/cyclin E and CDK5/cyclin/p35 (IC50 values are 0.68, 7.5 and 0.85 μM respectively). Selec
SMLES: BrC1=CC=C2NC3=C(CC(NC4=CC=CC=C34)=O)C2=C1
CAS NO: 760981-83-7
Standard In CHIKey: QQUXFYAWXPMDOE-UHFFFAOYSA-NAdrenergic Receptor inhibitors
Standard InChI: InChI=1S/C16H11BrN2O/c17-9-5-6-14-11(7-9)12-8-15(20)18-13-4-2-1-3-10(13)16(12)19-14/h1-7,19H,8H2,(H,18,20)
Typrof Compound:
Appearance:
Formula: C16H11BrN2O
M.Wt: 327.18
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/260/2/742
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in DMSO and to 5 mM in ethanol with gentle warming
Storage: Store at RT
Purity: >98%
Chemical Name: 9-Bromo-7,12-dihydro-indolo[3,2-d][1]benzazepin-6(5H)-one