Product Name: LE 300
Subtitle:
Biological Activity: Biological Activity of LE 300Potent and selective dopamine D1 receptor antagonist (Ki values are 0.08 – 1.9 nM and 6 – 45 nM for D1 and D2 receptors respectively). Also displays moderate affinity for the 5-HT2A receptor (Ki = 20 nM). Active in vivo.
SMLES: CN1CCC2=C(CC3=CC=CC=C3CC1)NC4=CC=CC=C24
CAS NO: 15176-29-1
Standard In CHIKey: Somatostatin Receptor inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C20H22N2
M.Wt: 290.41
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/270/1/77
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 50 mM in 1eq. HCl and to 100 mM in DMSO
Storage: Store at RT
Purity: >98%
Chemical Name: 6,7,8,9,14,15-Hexahydro-7-methyl-5H-indolo[3,2-f][3]benzazecine