Product Name: Mepyramine maleate
Subtitle:
Biological Activity: Biological Activity of Mepyramine maleateSelective inverse agonist for the H1 receptor. Inhibits histamine induced inositol phosphate (InsP) production (log EC50 = -7.94) and intracellular calcium mobilization. Sequesters Gq/11 protein, reducing its avail
SMLES: CN(C)CCN(C1=NC=CC=C1)CC(C=C2)=CC=C2OC.OC(/C=CC(O)=O)=O
CAS NO: 38821-53-3
Standard In CHIKey: JXYWFNAQESKDNC-BTJKTKAUSA-NDNA-PK inhibitors
Standard InChI: InChI=1S/C17H23N3O.C4H4O4/c1-19(2)12-13-20(17-6-4-5-11-18-17)14-15-7-9-16(21-3)10-8-15;5-3(6)1-2-4(7)8/h4-11H,12-14H2,1-3H3;1-2H,(H,5,6)(H,7,8)/b;2-1-
Typrof Compound:
Appearance:
Formula: C17H23N3O.C4H4O4
M.Wt: 401.46
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/269/3/948
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in water and to 100 mM in DMSO
Storage: Store at RT
Purity: >98%
Chemical Name: 2-((2-(Dimethylamino)ethyl)(p-methoxybenzyl)amino)-pyridine maleate