Product Name: P1075
Subtitle:
Biological Activity: Biological Activity of P1075Potent Kir6 (KATP) channel opener (EC50 for relaxation of rat aorta = 7.5 nM). Binds to SUR2A and SUR2B with high affinity (Kd values are 17 and 3 nM respectively).
SMLES: N#CN/C(NC1=CC=CN=C1)=NC(C)(C)CC
CAS NO: 6880-91-7
Standard In CHIKey: HKZNADVVGXKQDL-UHFFFAOYSA-NPhosphodiesterase PDE) inhibitors
Standard InChI: InChI=1S/C12H17N5/c1-4-12(2,3)17-11(15-9-13)16-10-6-5-7-14-8-10/h5-8H,4H2,1-3H3,(H2,15,16,17)
Typrof Compound:
Appearance:
Formula: C12H17N5
M.Wt: 231.3
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/273/3/1015
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 50 mM in ethanol and to 100 mM in DMSO
Storage: Store at RT
Purity: >98%
Chemical Name: N-cyano-N-(1,1-dimethylpropyl)-N-3-pyridylguanidine