Product Name: PHP 501 trifluoroacetate
Subtitle:
Biological Activity: Biological Activity of PHP 501 trifluoroacetatePotent GABAA antagonist (Ki = 0.0028 μM at rat GABAA receptors; IC50 = 0.024 μM at human α1β2γ2 GABAA-expressing tsA201 cells). Displays no inhibitory activity at hGAT-1, hGAT-2, hGAT
SMLES: N/A
CAS NO: 890643-16-0
Standard In CHIKey: SRPK inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C20H21N3O.CF3CO2H
M.Wt: 433.42
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/272/3/1011
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in DMSO
Storage: Store at -20℃
Purity: >98%
Chemical Name: 4-(5-[1,1-Biphenyl]-3-yl-1-hydroxy-1H-pyrazol-4-yl)piperidine trifluoroacetate