Product Name: PK 44 phosphate
Subtitle: DPP-IV inhibitor
Biological Activity: Biological Activity of PK 44 phosphateDescription PK 44 phosphate is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV) with an IC50 value of 15.8 nM. Targets DPP-IV IC50 15.8 nM
SMLES: O=C(N1CC2=NN=C(C(F)(F)F)N2CC1)C[C@H](N)CC3=NNC4=C3C=CC(F)=C4F.O=P(O)(O)O
CAS NO: 30220-46-3
Standard In CHIKey: CETP inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C17H16F5N7O.H3PO4
M.Wt: 527.34
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/271/2/708
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: (R)-3-amino-4-(6,7-difluoro-1H-indazol-3-yl)-1-(3-(trifluoromethyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)butan-1-one phosphate