Product Name: (S)-WAY 100135 dihydrochloride
Subtitle: 5-HT1A receptor antagonist,potent and selective
Biological Activity: Biological Activity of (S)-WAY 100135 dihydrochloridePotent, selective 5-HT1A receptor antagonist (IC50 = 15 nM). Selective over 5-HT1B, 1C, 2,α1, α2 and D2 receptors (IC50 > 1000 nM). Centrally active on systemic administration.
SMLES: CN1N=C(N=N1)C2=NC=C(C=C2)C3=C(C=C(C=C3)N4CC(OC4=O)CO)F
CAS NO: 132-98-9
Standard In CHIKey: GPR139 inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C24H33N3O2.2HCl
M.Wt: 468.47
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/270/1/285
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in DMSO and to 5 mM in water with gentle warming and to 10 mM in water with sonication
Storage: Desiccate at +4℃
Purity: >98%
Chemical Name: (S)-N-tert-Butyl-3-(4-(2-methoxyphenyl)-piperazin-1-yl)-2-phenylpropanamide dihydrochloride