Product Name: SB 204741
Subtitle:
Biological Activity: Biological Activity of SB 204741Potent and selective 5-HT2B receptor antagonist (pA2 = 7.95). Displays ≥ 135-fold selectivity over 5-HT2C (pKi = 5.82), 5-HT2A (pKi < 5.2), 5-HT1A, 1D, 1E, 5-HT3 and 5-HT4 receptors.
SMLES: O=C(NC1=CC(C)=NS1)NC2=CC=C3N(C)C=CC3=C2
CAS NO: 122628-50-6
Standard In CHIKey: HCN Channel inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C14H14N4OS
M.Wt: 286.35
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/265/1/248
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in DMSO and to 20 mM in ethanol
Storage: Store at RT
Purity: >98%
Chemical Name: N-(1-Methyl-1H-indolyl-5-yl)-N-(3-methyl-5-isothiazolyl)urea