Product Name: SB 452533
Subtitle:
Biological Activity: Biological Activity of SB 452533Potent TRPV1 antagonist against capsaicin (pKb = 7.7), noxious heat and acid-mediated (pIC50 = 7.0) receptor activation (pKi = 6.22 at the recombinant hTRPV1 receptor). Exhibits analgesic properties.
SMLES: N/A
CAS NO: 1253186-49-0
Standard In CHIKey: Arenavirus inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C18H22BrN3O
M.Wt: 376.29
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/274/1/72
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in DMSO and to 10 mM in ethanol with gentle warming
Storage: Store at RT
Purity: >98%
Chemical Name: N-(2-Bromophenyl)-N-[2-[ethyl(3-methylphenyl)amino]ethyl]-urea