Product Name: SKF 89976A hydrochloride
Subtitle:
Biological Activity: Biological Activity of SKF 89976A hydrochlorideA potent GABA uptake inhibitor, selective for GAT-1 (IC50 values are 0.13, 550, 944 and 7210 μM for hGAT-1, rGAT-2, hGAT-3 and hBGT-1 respectively). Inhibits transport current competitively (Ki = 7 μM)
SMLES: OC([C@H]1CN(CC/C=C(C2=CC=CC=C2)/C3=CC=CC=C3)CCC1)=O.Cl
CAS NO: 959746-77-1
Standard In CHIKey: Cathepsin inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C22H25NO2.HCl
M.Wt: 371.91
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/273/2/734
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in water with gentle warming and to 100 mM in DMSO
Storage: Desiccate at +4℃
Purity: >98%
Chemical Name: 1-(4,4-Diphenyl-3-butenyl)-3-piperidinecarboxylic acid hydrochloride