Product Name: TC-G 1004
Subtitle:
Biological Activity: Biological Activity of TC-G 1004Potent antagonist of adenosine A2A receptors; displays >100-fold selectivity for A2A over A1 receptors (Ki values are 0.44 and 85 nM respectively). Potentiates L-DOPA-induced rotational behavior in 6-OHDA-lesioned rats
SMLES: O=C(C)NC1=CC(C2=CC=CC(N3CCC(CC3)OC)=N2)=NC(N4N=C(C)C=C4C)=N1
CAS NO: 870093-23-5
Standard In CHIKey: Bcl-2 Family inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C22H27N7O2
M.Wt: 421.5
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/264/1/489
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in 1eq. HCl and to 100 mM in DMSO
Storage: Store at -20℃
Purity: >98%
Chemical Name: N-[2-(3,5-Dimethyl-1H-pyrazol-1-yl)-6-[6-(4-methoxy-1-piperidinyl)-2-pyridinyl]-4-pyrimidinyl]acetamide