Product Name: TG100713
Subtitle: pan-PI3K inhibitor
Biological Activity: Biological Activity of TG100713Inhibitor of PI3-kinase (IC50 values are 24, 50, 165 and 215 nM for PI3Kδ, γ, α and β isoforms respectively). Inhibits endothelial cell proliferation.
SMLES: C1=CC(=CC(=C1)O)C2=CN=C3C(=N2)C(=NC(=N3)N)N
CAS NO: 104376-79-6
Standard In CHIKey: P2Y Receptor inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C12H10N6
M.Wt: 254.25
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/271/1/238
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 10 mM in DMSO
Storage: Desiccate at RT
Purity: >98%
Chemical Name: 3-(2,4-Diamino-6-pteridinyl)-phenol