Product Name: YM201636
Subtitle: PIKfyve inhibitor,potent and selective
Biological Activity: Biological Activity of YM201636Description YM201636 is a selective inhibitor of PIKfyve with an IC50 value of 33 nM. Targets PIKfyve p110α IC50 33 nM 3.3 μM
SMLES: C1COCCN1C2=NC(=NC3=C2OC4=C3C=CC=N4)C5=CC(=CC=C5)NC(=O)C6=CN=C(C=C6)N
CAS NO: 67-20-9
Standard In CHIKey: Immunology_Inflammation inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C25H21N7O3
M.Wt: 467.48
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/271/1/302
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: 6-amino-N-[3-(4-morpholin-4-ylpyrido[2,3]furo[2,4-b]pyrimidin-2-yl)phenyl]pyridine-3-carboxamide