Product Name :
Azatadine dimaleate
Synonym :
6,11-Dihydro-11-(1-methyl-4-piperidinylidene)-5H-benzo[5,6]cyclohepta[1,2-b]pyridineAzatadine Dimaleate
Chemical Name :
CAS NO.:
3978-86-7
Molecular formula :
C20H22N2·2C4H4O4
Molecular Weight:
522.55 g/mol
Classification :
MedChemExpress Products > Research Chemicals >Fine Chemicals > Azatadine dimaleate
Description:
Azatadine is an antihistamine that has been shown to be clinically relevant for the treatment of allergic symptoms. Azatadine has been shown to bind to voltage-dependent calcium channels and inhibit their opening, preventing the release of neurotransmitters such as acetylcholine. Azatadine also blocks leukotriene receptors and therefore its activity is antagonistic with fatty acid synthase inhibitors and other pharmacological agents.Azatadine dimaleate (AZA) is a prodrug that is metabolized in vivo by esterases into the active form, azatadine. AZA inhibits histamine release from mast cells in vitro and in vivo models. This drug also has anti-inflammatory properties that may be due to its inhibition of prostaglandin synthesis.
Purity :
>98%
Specifications :
10 mM * 1 mL
Price.:
66
Price unit :
$
Inventory :
In stock
Related websites: https://www.medchemexpress.com
587871-26-9 References 83905-01-5 Molecular Weight PMID:25905294 MedChemExpress (MCE) offers a wide range of high-quality research chemicals and biochemicals (novel life-science reagents, reference compounds and natural compounds) for scientific use. We have professionally experienced and friendly staff to meet your needs. We are a competent and trustworthy partner for your research and scientific projects.Related websites: https://www.medchemexpress.com