Product Name: ENMD-2076
Subtitle: Selective Aurora A/Flt3 inhibitor
Biological Activity: Biological Activity of ENMD-2076Description ENMD-2076 is a selective inhibitor of Aurora A and Flt3 with IC50 values of 14 nM and 1.86 nM, respectively. Targets Aurora A Flt3 IC50 14 nM 1.86 nM
SMLES: CC1=CC(=NN1)NC2=NC(=NC(=C2)N3CCN(CC3)C)C=CC4=CC=CC=C4
CAS NO: 171335-80-1
Standard In CHIKey: Sigma Receptor inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C21H25N7
M.Wt: 375.47
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/253/3/1002
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: 6-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)-2-[(E)-2-phenylethenyl]pyrimidin-4-amine