Product Name: MRS 1334
Subtitle:
Biological Activity: Biological Activity of MRS 1334Potent and highly selective antagonist for the human adenosine A3 receptor. Ki values are 2.69 nM at hA3, and > 100 μM at rat A1 and rat A2A receptors.
SMLES: O=C(C1=C(C2=CC=CC=C2)NC(C)=C(C(OCC)=O)[C@H]1C#CC3=CC=CC=C3)OCC4=CC=CC([N+]([O-])=O)=C4
CAS NO: 460746-46-7
Standard In CHIKey: Pyruvate Dehydrogenase inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C31H26N2O6
M.Wt: 522.56
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/263/2/682
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in DMSO
Storage: Desiccate at -20℃
Purity: >98%
Chemical Name: 1,4-Dihydro-2-methyl-6-phenyl-4-(phenylethynyl)-3,5-pyridinedicarboxylic acid 3-ethyl-5-[(3-nitrophenyl)methyl] ester