Product Name: PHA-767491
Subtitle: Cdc7/cdk9 inhibitor, potent, ATP-competitive
Biological Activity: Biological Activity of PHA-767491Description PHA-767491 is a potent, ATP-competitive inhibitor of cdc7 and cdk9 with 10 nM and 34 nM, respectively. Targets cdc7 cdk9 IC50 10 nM 34 nM
SMLES: C1CNC(=O)C2=C1NC(=C2)C3=CC=NC=C3
CAS NO: 923604-59-5
Standard In CHIKey: CETP inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C12H11N3O
M.Wt: 213.24
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/252/1/159
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: 2-pyridin-4-yl-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-one