Product Name: PHA-793887
Subtitle: Pan-Cdk inhibitor
Biological Activity: Biological Activity of PHA-793887Description PHA-793887 is a novel and potent inhibitor of CDK2, CDK5 and CDK7 with IC50 values of 8 nM, 5 nM and 10 nM, respectively. Targets CDK5/p25 CDK2/CyclinA CDK2/CyclinE CDK7/CyclinH CDK1/CyclinB I
SMLES: CC(C)CC(=O)NC1=NNC2=C1CN(C2(C)C)C(=O)C3CCN(CC3)C
CAS NO: 60940-34-3
Standard In CHIKey: Glucokinase inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C19H31N5O2
M.Wt: 361.48
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/252/1/253
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: N-[6,6-dimethyl-5-(1-methylpiperidine-4-carbonyl)-1,4-dihydropyrrolo[3,4-c]pyrazol-3-yl]-3-methylbutanamide