Product Name: TAK-875
Subtitle: GPR40 agonist
Biological Activity: Biological Activity of TAK-875Description TAK-875 is a selective agonist of GPR40 with EC50 of 14 nM, 400-fold more potent than oleic acid. Targets GPR40 IC50 14 nM (EC50)
SMLES: CC1=CC(=CC(=C1C2=CC(=CC=C2)COC3=CC4=C(C=C3)C(CO4)CC(=O)O)C)OCCCS(=O)(=O)C
CAS NO: 737727-12-7
Standard In CHIKey: PKD inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C29H32O7S
M.Wt: 524.64
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/262/1/398
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: 2-[(3S)-6-[[3-[2,6-dimethyl-4-(3-methylsulfonylpropoxy)phenyl]phenyl]methoxy]-2,3-dihydro-1-benzofuran-3-yl]acetic acid