Product Name: RI-1Subtitle: RAD51 inhibitor,cell-permeableBiological Activity: Biological Activity of RI-1Description RI-1 is a cell-permeable inhibitor of RAD51. Targets RAD51 IC50SMLES: C1COCCN1C2=C(C(=O)N(C2=O)C3=CC(=C(C=C3)Cl)Cl)ClCAS NO: 912445-05-7Standard In CHIKey: DGAT inhibitorsStandard InChI: Typrof Compound:…
Product Name: PyridostatinSubtitle: Drug used for promoting growth arrestBiological Activity: SMLES: C1=CC=C2C(=C1)C(=CC(=N2)NC(=O)C3=CC(=CC(=N3)C(=O)NC4=NC5=CC=CC=C5C(=C4)OCCN)OCCN)OCCNCAS NO: 229975-97-7Standard In CHIKey: Cytochrome P450 inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C31H32N8O5M.Wt: 596.64General Tips: For obtaining a…
Product Name: PoloxinSubtitle: PLK1 inhibitorBiological Activity: SMLES: CC1=CC=CC=C1C(=O)ON=C2C=C(C(=O)C=C2C)C(C)CCAS NO: 1005342-46-0Standard In CHIKey: COMT inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C18H19NO3M.Wt: 297.35General Tips: For obtaining a higher solubility , please warm…
Product Name: PHA-767491Subtitle: Cdc7/cdk9 inhibitor, potent, ATP-competitiveBiological Activity: Biological Activity of PHA-767491Description PHA-767491 is a potent, ATP-competitive inhibitor of cdc7 and cdk9 with 10 nM and 34 nM, respectively. Targets…
Product Name: PF-3758309Subtitle: PAK4 inhibitorBiological Activity: Biological Activity of PF-3758309Description PF-03758309 is a potent, ATP-competitive, pyrrolopyrazole inhibitor of PAK4 with IC50 of 1.3 nM. Targets PAK4 IC50 Ki=18.7 nM, Kd…
Product Name: NVP-LCQ195Subtitle: CDK1/CDK2/CDK5 inhibitorBiological Activity: SMLES: O=S(=O)(N3CCC(NC(=O)c2c(NC(=O)c1c(Cl)cccc1Cl)cnn2)CC3)CCAS NO: 302962-49-8Standard In CHIKey: Carboxypeptidase inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C17H19Cl2N5O4SM.Wt: 460.33General Tips: For obtaining a higher solubility , please warm…
Product Name: Monomethyl auristatin ESubtitle: Antimitotic agentBiological Activity: Biological Activity of Monomethyl auristatin EPotent, synthetic, cytotoxic analog of dolastatin 10. Suppresses tumor cell viability in vitro (GIC50 values are 0.22,…
Product Name: MMADSubtitle: Tubulin inhibitor,highly potentBiological Activity: Biological Activity of MMADDescription Monomethyl auristatin D (MMAD) is a potent inhibitor of tubulin. Targets tubulin ADCs toxin IC50SMLES: O=C(((OC)1()CCCN1C(C(OC)(N(C)C((NC((C(C)C)N()C)=O)C(C)C)=O)(C)CC)=O)C)N(C2=NC=CS2)CC3=CC=CC=C3CAS NO: 585543-15-3Standard In…
Product Name: Mc-MMADSubtitle: Potent tubulin inhibitorBiological Activity: SMLES: CC(CCC(C1CC1)O)C2CCC3C2(CCCC3=CC=C4CC(CC(C4=C)O)O)CCAS NO: 1421373-66-1Standard In CHIKey: ATGL inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C51H77N7O9SM.Wt: 964.26General Tips: For obtaining a higher solubility , please…
Product Name: LY2835219 free baseSubtitle: CDK inhibitorBiological Activity: SMLES: CCN1CCN(CC1)Cc2ccc(nc2)Nc3ncc(c(n3)c4cc5c(c(c4)F)nc(n5C(C)C)C)FCAS NO: 1218778-77-8Standard In CHIKey: Angiotensin-converting Enzyme ACE) inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C27H32F2N8M.Wt: 506.59General Tips: For obtaining a higher…