Product Name: 2-Furoyl-LIGRLO-amideSubtitle: Biological Activity: Biological Activity of 2-Furoyl-LIGRLO-amidePotent and selective PAR2 receptor agonist (pD2 = 7.0). Causes a dose-dependent relaxation of murine femoral arteries.SMLES: N/ACAS NO: 851546-61-7Standard In CHIKey:…
Product Name: TRAP-6Subtitle: PAR1 agonistBiological Activity: Biological Activity of TRAP-6Peptide fragment (residues 42-47) of protease-activated receptor 1 (PAR1) that acts as a PAR1 agonist. Stimulates platelet aggregation (EC50 = 0.8…
Product Name: PAR 4 (1-6)Subtitle: PAR4 agonistBiological Activity: SMLES: N/ACAS NO: 1523406-39-4Standard In CHIKey: mGluR inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C28H41N7O9M.Wt: 619.68General Tips: For obtaining a higher solubility ,…
Product Name: LRGILS-NH2Subtitle: Biological Activity: Biological Activity of LRGILS-NH2Reversed amino acid sequence control peptide for SLIGRL-NH2, a protease-activated receptor-2 (PAR2) agonist that facilitates gastrointestinal transit in vivo.SMLES: N/ACAS NO: 1373423-53-0Standard…
Product Name: RLLFT-NH2Subtitle: Biological Activity: Biological Activity of RLLFT-NH2Reversed amino acid sequence control peptide for TFLLR-NH2, a PAR1 selective agonist that significantly increases nociceptive threshold.SMLES: CC(C)CC(C(=O)NC(CC(C)C)C(=O)NC(CC1=CC=CC=C1)C(=O)NC(C(C)O)C(=O)N)NC(=O)C(CCCN=C(N)N)NCAS NO: 1448347-49-6Standard In CHIKey:…
Product Name: VKGILS-NH2Subtitle: control peptide for SLIGKV-NH2, PAR1 agonistBiological Activity: Biological Activity of VKGILS-NH2Reversed amino acid sequence control peptide for SLIGKV-NH2, a protease-activated receptor 2 (PAR2) agonist.SMLES: CC((/N=C(O)/C/N=C(O)/(/N=C(O)/(N)()C(C)C)()CCCCN)()/C(O)=N/(/C(O)=N/(C(O)=N)()CO)()CC(C)C)()CCAS NO: 53123-88-9Standard…
Product Name: AC 264613Subtitle: PAR2 agonist,potent and selectiveBiological Activity: Biological Activity of AC 264613Potent and selective protease-activated receptor 2 (PAR2) agonist (pEC50 = 7.5). Displays no activity at other PAR…
Product Name: AC 55541Subtitle: PAR2 agonist,potent and selectiveBiological Activity: Biological Activity of AC 55541Potent and selective protease-activated receptor 2 (PAR2) agonist (pEC50 = 6.7) that displays no activity at other…
Product Name: Thrombin Receptor Agonist PeptideSubtitle: Biological Activity: Biological Activity of Thrombin Receptor Agonist PeptideAgonist at the thrombin receptor; causes platelet aggregation (EC50 = 4 μM) and secretion.SMLES: CC(C)CC(C(=O)NC(CC(C)C)C(=O)NC(CCCNC(=N)N)C(=O)NC(CC(=O)N)C(=O)N1CCCC1C(=O)NC(CC(=O)N)C(=O)NC(CC(=O)O)C(=O)NC(CCCCN)C(=O)NC(CC2=CC=C(C=C2)O)C(=O)NC(CCC(=O)O)C(=O)N3CCCC3C(=O)NC(CC4=CC=CC=C4)C(=O)O)NC(=O)C(CC5=CC=CC=C5)NC(=O)C(CO)NCAS NO:…
Product Name: AY-NH2Subtitle: Selective PAR4 agonistBiological Activity: Biological Activity of AY-NH2Selective PAR4 receptor agonist peptide. Stimulates platelet aggregation in vitro (EC50 = 15 μM). Exhibits an increase in paw thickness…