Product Name: MDV3100 (Enzalutamide)
Subtitle: Androgen receptor antagonist
Biological Activity: Biological Activity of MDV3100 (Enzalutamide)Description Enzalutamide (MDV3100) is an antagonist of androgen-receptor (AR) with IC50 of 36 nM. Targets Androgen-receptor IC50 36 nM
SMLES: CC1(C(=O)N(C(=S)N1C2=CC(=C(C=C2)C(=O)NC)F)C3=CC(=C(C=C3)C#N)C(F)(F)F)C
CAS NO: 405098-33-1
Standard In CHIKey: CMV inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C21H16F4N4O2S
M.Wt: 464.4
General Tips: for obtaining a higher concentration: Please warm the tube at 37 °C for 10 minutes and/or shake it in the ultrasonic bath for a while.Stock solution can be stored below -20°C for several months.PubMed ID:http://jpet.aspetjournals.org/content/252/3/929
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: 4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluoro-N-methylbenzamide