Product Name: UNC0638
Subtitle: G9a/GLP HMTase inhibitor, potent and selective
Biological Activity: Biological Activity of UNC0638Description UNC0638 is a potent and selective inhibitor of G9a and GLP HMTase with IC50 values of < 15 nM and 19 nM, respectively. Targets G9a GLP IC50 < 15 nM 19 nM
SMLES: CC(C)N1CCC(CC1)Nc2c3cc(c(cc3nc(n2)C4CCCCC4)OCCCN5CCCC5)OC
CAS NO: 736992-21-5
Standard In CHIKey: Adenosine Receptor inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C30H47N5O2
M.Wt: 509.72
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/253/2/537
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: 2-Cyclohexyl-N-(1-isopropyl-4-piperidinyl)-6-methoxy-7-[3-(1-pyrrolidinyl)propoxy]-4-quinazolinamine