Product Name: SGC-CBP30
Subtitle: Inhibitor of CREBBP/EP300 bromodomain,potent
Biological Activity: Biological Activity of SGC-CBP30Description SGC-CBP30 is a potent inhibitor of CREBBP/EP300 with IC50 values of 21 nM and 38 nM, respectively. Targets CREBBP EP300 IC50 21 nM 38 nM
SMLES: CC1=C(C(=NO1)C)C2=CC3=C(C=C2)N(C(=N3)CCC4=CC(=C(C=C4)OC)Cl)CC(C)N5CCOCC5
CAS NO: 670220-88-9
Standard In CHIKey: Chloride Channel inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C28H33ClN4O3
M.Wt: 509.04
General Tips: for obtaining a higher concentration: Please warm the tube at 37 ℃ for 10 minutes and/or shake it in the ultrasonic bath for a while. Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/253/3/1265
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: 4-[(2S)-1-[2-[2-(3-chloro-4-methoxyphenyl)ethyl]-5-(3,5-dimethyl-1,2-oxazol-4-yl)benzimidazol-1-yl]propan-2-yl]morpholine