Product Name: MTEP hydrochloride
Subtitle: MGlu5 antagonist
Biological Activity: Biological Activity of MTEP hydrochloridePotent, selective and non-competitive mGlu5 antagonist (IC50 = 5 nM in Ca2+-flux assay; Ki= 16 nM). Displays anxiolytic activity in vivo and is orally active.
SMLES: CC1=NC(=CS1)C#CC2=CN=CC=C2.Cl
CAS NO: 156161-89-6
Standard In CHIKey: Renin inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C11H9ClN2S
M.Wt: 236.72
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/254/2/383
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in water and to 100 mM in DMSO
Storage: Store at -20℃
Purity: >98%
Chemical Name: 3-((2-Methyl-1,3-thiazol-4-yl)ethynyl)pyridine hydrochloride