Product Name: WZ811
Subtitle: Competitive CXCR4 antagonist,highly potent
Biological Activity: Biological Activity of WZ811Potent chemokine receptor type 4 (CXCR4) antagonist (EC50 = 0.3 nM). Inhibits CXCR4/stromal cell-derived factor-1 (SDF-1)-mediated modulation of cAMP in vitro (EC50 = 1.2 nM).
SMLES: C1=CC=NC(=C1)NCC2=CC=C(C=C2)CNC3=CC=CC=N3
CAS NO: 223499-30-7
Standard In CHIKey: Histamine Receptor inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C18H18N4
M.Wt: 290.36
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/262/3/1154
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 25 mM in DMSO
Storage: Store at -20℃
Purity: >98%
Chemical Name: N1,N4-Di-2-pyridinyl-1,4-benzenedimethanamine