Product Name: BMS 182874 hydrochloride
Subtitle: ETA antagonist
Biological Activity: Biological Activity of BMS 182874 hydrochloridePotent, selective and competitive non-peptide endothelin ETA receptor antagonist (Ki = 48 nM). Displays > 1000-fold selectivity over ETB receptors. Inhibits ET-1-induced pressor response following oral or
SMLES:
CAS NO: 1820565-69-2
Standard In CHIKey: SGK inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C17H19N3O3S.HCl
M.Wt: 381.88
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/263/2/708
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in DMSO
Storage: Store at RT
Purity: >98%
Chemical Name: 5-(Dimethylamino)-N-(3,4-dimethyl-5-isoxazolyl)-1-naphthalenesulfonamide hydrochloride