Product Name: TaranabantSubtitle: Biological Activity: SMLES: CC(C(CC1=CC=C(C=C1)Cl)C2=CC=CC(=C2)C#N)NC(=O)C(C)(C)OC3=NC=C(C=C3)C(F)(F)FCAS NO: 1374516-07-0Standard In CHIKey: ADC Cytotoxin inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C27H25ClF3N3O2M.Wt: 515.97General Tips: For obtaining a higher solubility , please warm…
Product Name: Talnetant hydrochlorideSubtitle: NK3 receptor antagonistBiological Activity: SMLES: CCC(C1=CC=CC=C1)NC(=O)C2=C(C(=NC3=CC=CC=C32)C4=CC=CC=C4)O.ClCAS NO: 173865-33-3Standard In CHIKey: BHCSUEHQURQVLD-BDQAORGHSA-NAntibody-drug Conjugate_ADC Related inhibitorsStandard InChI: InChI=1S/C25H22N2O2.ClH/c1-2-20(17-11-5-3-6-12-17)27-25(29)22-19-15-9-10-16-21(19)26-23(24(22)28)18-13-7-4-8-14-18;/h3-16,20,28H,2H2,1H3,(H,27,29);1H/t20-;/m0./s1Typrof Compound: Appearance: Formula: C25H23ClN2O2M.Wt: 418.92General Tips: For obtaining a higher…
Product Name: TalnetantSubtitle: NK3 receptor antagonist,potent and selectiveBiological Activity: Biological Activity of TalnetantPotent and selective non-peptide NK3 receptor antagonist (Ki values are 1, 144 and >100000 nM for human NK3,…
Product Name: Cerdulatinib (PRT062070)Subtitle: Syk/JAK inhibitorBiological Activity: SMLES: NC(C1=CN=C(NC2=CC=C(N3CCN(S(=O)(CC)=O)CC3)C=C2)N=C1NC4CC4)=OCAS NO: 1110766-97-6Standard In CHIKey: RSV inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C20H27N7O3SM.Wt: 445.54General Tips: for obtaining a higher concentration: Please warm…
Product Name: UNC 0642Subtitle: G9a and GLP histone lysine methyltransferase inhibitorBiological Activity: Biological Activity of UNC 0642Potent and selective G9a and GLP histone lysine methyltransferase inhibitor (IC50 < 2.5 nM).…
Product Name: C 21Subtitle: Protein arginine methyltransferase 1 (PRMT1) inhibitorBiological Activity: Biological Activity of C 21Selective protein arginine methyltransferase 1 (PRMT1) inhibitor (IC50 = 1.8 μM). Exhibits five-fold selectivity for…
Product Name: TC-E 5003Subtitle: PRMT1 inhibitor, potentBiological Activity: Biological Activity of TC-E 5003Selective protein arginine methyltransferase 1 (PRMT1) inhibitor (IC50 = 1.5 μM); exhibits no inhibitory activity against CARM1 and…
Product Name: L002Subtitle: Biological Activity: Biological Activity of L002p300 inhibitor (IC50 = 1.98 μM). Inhibits histone and p53 acetylation, and suppresses STAT3 activation in cell-based assays. Also suppresses tumor growth…
Product Name: (R)-(+)-Etomoxir sodium saltSubtitle: Biological Activity: Biological Activity of (R)-(+)-Etomoxir sodium saltInhibitor of carnitine palmitoyltransferase I (CPT1); inhibits β-oxidation in mitochondria. Shown to inhibit cardiolipin biosynthesis from exogenous fatty…
Product Name: Tranylcypromine hydrochlorideSubtitle: Biological Activity: Biological Activity of Tranylcypromine hydrochlorideIrreversible inhibitor of lysine-specific demethylase 1 (LSD1/BHC110) and monoamine oxidase (MAO). Inhibits histone demethylation. In combination with CHIR 99021, enables…