GSK2801
Product Name: GSK2801Subtitle: inhibitor of BAZ2A and BAZ2B bromodomainsBiological Activity: Biological Activity of GSK2801Selective BAZ2A and BAZ2B inhibitor (IC50 values are 0.40 and 0.43 μM, respectively). Selective for BAZ2A/B over…
PFI 4
Product Name: PFI 4Subtitle: Potent and selective BRPF1 Bromodomain inhibitorBiological Activity: Biological Activity of PFI 4Potent and selective BRPF1 bromodomain inhibitor (IC50 = 80 nM). Exhibits >100-fold selectivity for BRPF1…
2,4-Pyridinedicarboxylic Acid
Product Name: 2,4-Pyridinedicarboxylic AcidSubtitle: Histone LSD inhibitorBiological Activity: SMLES: O=C(O)C1=CC(C(O)=O)=NC=C1CAS NO: 473-98-3Standard In CHIKey: MJIVRKPEXXHNJT-UHFFFAOYSA-NSteroids inhibitorsStandard InChI: InChI=1S/C7H5NO4/c9-6(10)4-1-2-8-5(3-4)7(11)12/h1-3H,(H,9,10)(H,11,12)Typrof Compound: Appearance: Formula: C7H5NO4M.Wt: 167.12General Tips: For obtaining a higher solubility ,…
Triacetyl Resveratrol
Product Name: Triacetyl ResveratrolSubtitle: Cell-permeable resveratrol prodrugBiological Activity: SMLES: CC(OC1=CC=C(C=C1)/C()=C()/C2=CC(OC(C)=O)=CC(OC(C)=O)=C2)=OCAS NO: 520-34-3Standard In CHIKey: Flavonoids inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C20H18O6M.Wt: 354.35General Tips: For obtaining a higher solubility ,…
Sanguinarine chloride
Product Name: Sanguinarine chlorideSubtitle: Inhibitor of PP2C and MKP-1Biological Activity: Biological Activity of Sanguinarine chlorideInhibitor of protein phosphatase 2C (PP2C), selective over PP1, PP2A and PP2B in vitro. Also inhibits…
2-hexyl-4-Pentynoic Acid
Product Name: 2-hexyl-4-Pentynoic AcidSubtitle: Potent and robust HDACs inhibitorBiological Activity: SMLES: CCCCCCC(C(O)=O)CC#CCAS NO: Standard In CHIKey: DUQSBRQHALCSLC-UHFFFAOYSA-NPhenylpropanoids inhibitorsStandard InChI: InChI=1S/C11H18O2/c1-3-5-6-7-9-10(8-4-2)11(12)13/h2,10H,3,5-9H2,1H3,(H,12,13)Typrof Compound: Appearance: Formula: C11H18O2M.Wt: 182.26General Tips: For obtaining a higher…
BML-210(CAY10433)
Product Name: BML-210(CAY10433)Subtitle: Novel HDAC inhibitorBiological Activity: SMLES: CAS NO: 1668565-74-9Standard In CHIKey: Saccharides and Glycosides inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C20H25N3O2M.Wt: 339.43General Tips: For obtaining a higher solubility…
UF 010
Product Name: UF 010Subtitle: Novel and selective class I HDAC inhibitorBiological Activity: Biological Activity of UF 010Class I HDAC inhibitor (IC50 values are 0.06, 0.1, 0.5 and 1.5 μM for…
BG45
Product Name: BG45Subtitle: Novel HDAC3-selective inhibitorBiological Activity: SMLES: CAS NO: 162411-29-2Standard In CHIKey: Cell_Counting_Kit-8 inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C11H10N4OM.Wt: 214.22General Tips: For obtaining a higher solubility , please…
ACY-241
Product Name: ACY-241Subtitle: Selective and orally active HDAC6 inhibitorBiological Activity: SMLES: CAS NO: 75350-46-8Standard In CHIKey: Phosphatase_Inhibitor_Cocktail_III inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C24H26ClN5O3M.Wt: 467.95General Tips: For obtaining a higher…