Product Name: EtomoxirSubtitle: (CPT)-1 and DGAT activity inhibitorBiological Activity: SMLES: CCOC(=O)1(CO1)CCCCCCOC2=CC=C(C=C2)ClCAS NO: 552325-16-3Standard In CHIKey: DZLOHEOHWICNIL-KRWDZBQOSA-NGPCR19 inhibitorsStandard InChI: InChI=1S/C17H23ClO4/c1-2-20-16(19)17(13-22-17)11-5-3-4-6-12-21-15-9-7-14(18)8-10-15/h7-10H,2-6,11-13H2,1H3/t17-/m0/s1Typrof Compound: Appearance: Formula: C17H23ClO4M.Wt: 326.82General Tips: For obtaining a higher solubility…
Product Name: DMP 777Subtitle: Leukocyte elastase (HLE) inhibitorBiological Activity: SMLES: CCCC(C1=CC2=C(C=C1)OCO2)NC(=O)N3C(C(C3=O)(CC)CC)OC4=CC=C(C=C4)C(=O)N5CCN(CC5)CCAS NO: 873225-46-8Standard In CHIKey: ZSDCIRYNTCVTMF-GIGWZHCTSA-NGlucagon Receptor inhibitorsStandard InChI: InChI=1S/C31H40N4O6/c1-5-8-24(22-11-14-25-26(19-22)40-20-39-25)32-30(38)35-28(37)31(6-2,7-3)29(35)41-23-12-9-21(10-13-23)27(36)34-17-15-33(4)16-18-34/h9-14,19,24,29H,5-8,15-18,20H2,1-4H3,(H,32,38)/t24-,29+/m1/s1Typrof Compound: Appearance: Formula: C31H40N4O6M.Wt: 564.69General Tips: For obtaining a higher…
Product Name: DGAT-1 inhibitorSubtitle: Diacylglycerol acyltransferase (DGAT1) inhibitorBiological Activity: SMLES: CC1(C(=NC2=C(N=CN=C2O1)N)C3=CC=C(C=C3)C4CCC(CC4)CC(=O)O)CCAS NO: 1219168-18-9Standard In CHIKey: GHSR inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C22H26N4O3M.Wt: 394.2General Tips: For obtaining a higher solubility…
Product Name: DeltarasinSubtitle: KRAS-PDEδ interaction inhibitorBiological Activity: SMLES: CC(C)NC1=C(N=CC=C1)N2CCN(CC2)C(=O)C3=CC4=C(N3)C=CC(=C4)NS(=O)(=O)CCAS NO: 1446144-04-2Standard In CHIKey: Endothelin Receptor inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C40H37N5OM.Wt: 603.75General Tips: For obtaining a higher solubility ,…
Product Name: Bay 60-7550Subtitle: Potent PDE2 inhibitorBiological Activity: Biological Activity of Bay 60-7550Description Bay 60-7550 is a potent PDE2 inhibitor with IC50 values of 2.0 nM (bovine) and 4.7 nM…
Product Name: BalaglitazoneSubtitle: PPAR-γ partial agonistBiological Activity: Biological Activity of BalaglitazoneDescription Balaglitazone (DRF-2593; NN-2344) is a novel partial agonist of PPAR-γ. Targets PPARγ IC50SMLES: CAS NO: 453562-69-1Standard In CHIKey: Dopamine…
Product Name: AZD7687Subtitle: DGAT inhibitor,potent and selectiveBiological Activity: SMLES: CAS NO: 1300031-49-5Standard In CHIKey: CXCR inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C21H25N3O3M.Wt: 367.44General Tips: For obtaining a higher solubility ,…
Product Name: AN-2728Subtitle: PDE4 inhibitor,anti-inflammatory compoundBiological Activity: SMLES: CAS NO: 1187020-80-9Standard In CHIKey: CRTH2 GPR44) inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C14H10BNO3M.Wt: 251.05General Tips: For obtaining a higher solubility ,…
Product Name: AleglitazarSubtitle: PPARα/PPARγagonistBiological Activity: Biological Activity of AleglitazarDescription Aleglitazar (R1439) is a dual agonist of peroxisome proliferator-activated receptor (PPAR), with affinity to PPARα and PPARγ. Targets PPAR IC50SMLES: CAS…
Product Name: AGI-6780Subtitle: IDH2/R140Q mutation inhibitorBiological Activity: Biological Activity of AGI-6780Description AGI-6780 is a potent and time-dependent inhibitor of IDH2-R140Q with IC50 values of 23±1.7 nM and 190±8.1 nM for…