Product Name: AnisomycinSubtitle: JNK agonist, potent and specificBiological Activity: Biological Activity of AnisomycinProtein synthesis inhibitor (blocks translation). Potent activator of stress-activated protein kinases (JNK/SAPK) and p38 MAP kinase. Acts as…
Product Name: KT 5823Subtitle: Biological Activity: Biological Activity of KT 5823Selective inhibitor of protein kinase G (Ki values are 0.23, 4 and > 10 μM for inhibition of PKG, PKC…
Product Name: DEL-22379Subtitle: inhibitor of the dimerization of ERKBiological Activity: Biological Activity of DEL-22379ERK dimerization inhibitor (IC50 ~ 0.5 μM); inhibits ERK dimerization without effecting phosphorylation or kinase activity. Suppresses…
Product Name: BI-847325Subtitle: dual inhibitor of MEK and Aurora kinasesBiological Activity: SMLES: CAS NO: 38562-01-5Standard In CHIKey: Gap Junction Protein inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C29H28N4O2M.Wt: 464.56General Tips: For…
Product Name: Pexmetinib (ARRY-614)Subtitle: dual inhibitor of p38 MAPK and Tie2/Tek receptor tyrosine kinaseBiological Activity: SMLES: CC1=CC=C(N2C(N/C(O)=N/CC3=CC(F)=CC=C3OC4=CC=C5C(C=NN5CCO)=C4)=CC(C(C)(C)C)=N2)C=C1CAS NO: 1256580-46-7Standard In CHIKey: Dynamin inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C31H33FN6O3M.Wt: 556.63General…
Product Name: PF-03394197(Oclacitinib)Subtitle: Novel Janus kinase inhibitorBiological Activity: SMLES: CNS(C1()CC(N(C2=NC=NC3=C2C=CN3)C)()CC1)(=O)=OCAS NO: 1123838-51-6Standard In CHIKey: Arp2_3 Complex inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C15H23N5O2SM.Wt: 337.44General Tips: For obtaining a higher solubility…
Product Name: AS601245Subtitle: c-Jun NH2-terminal protein kinase inhibitorBiological Activity: SMLES: CAS NO: 606143-52-6Standard In CHIKey: Cytoskeleton inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C20H16N6SM.Wt: 372.45General Tips: For obtaining a higher solubility…
Product Name: RO5126766(CH5126766)Subtitle: Raf/MEK dual inhibitorBiological Activity: SMLES: CC(C1=C(O2)C=C(OC3=NC=CC=N3)C=C1)=C(C2=O)CC4=C(F)C(NS(NC)(=O)=O)=NC=C4CAS NO: 1232416-25-9Standard In CHIKey: Wee1 inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C21H18FN5O5SM.Wt: 471.46General Tips: For obtaining a higher solubility , please…
Product Name: GDC-0994Subtitle: ERK1/2 inhibitorBiological Activity: SMLES: CN1C(NC2=NC=CC(C(C=CN3(C4=CC(F)=C(Cl)C=C4)()CO)=CC3=O)=N2)=CC=N1CAS NO: 1629267-75-9Standard In CHIKey: Topoisomerase inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C21H18ClFN6O2M.Wt: 440.86General Tips: For obtaining a higher solubility , please warm…
Product Name: PD 334581Subtitle: Biological Activity: Biological Activity of PD 334581Inhibitor of MEK1. Analog of PD 184352.SMLES: N/ACAS NO: 747412-49-3Standard In CHIKey: Telomerase inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C20H19F3IN5O2M.Wt:…