Product Name: PD 334581Subtitle: Biological Activity: Biological Activity of PD 334581Inhibitor of MEK1. Analog of PD 184352.SMLES: N/ACAS NO: 747412-49-3Standard In CHIKey: Telomerase inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C20H19F3IN5O2M.Wt:…
Product Name: HI TOPK 032Subtitle: Biological Activity: Biological Activity of HI TOPK 032T-LAK-cell-originated protein kinase (TOPK) inhibitor; exhibits selectivity for TOPK over other MAPKK family members including ERK1, JNK1 and…
Product Name: PluripotinSubtitle: Biological Activity: SMLES: CC1=CC(=O)C2=C(C1=O)C=CC=C2OCAS NO: 779353-01-4Standard In CHIKey: Sirtuin inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C27H25F3N8O2M.Wt: 550.54General Tips: For obtaining a higher solubility , please warm the…
Product Name: PF-3644022Subtitle: Potent and Selective MK2 inhibitorBiological Activity: Biological Activity of PF-3644022Potent, ATP-competitive inhibitor of mitogen-activated protein kinase (MAPK)-activated protein kinase-2 (MK2) (IC50 = 5.2 nM; Ki = 3…
Product Name: AMG 548Subtitle: P38α inhibitor,potent and selectiveBiological Activity: Biological Activity of AMG 548Potent and selective inhibitor of p38α (Ki values are 0.5, 3.6, 2600 and 4100 nM for p38α,…
Product Name: JIP-1 (153-163)Subtitle: Biological Activity: Biological Activity of JIP-1 (153-163)Peptide inhibitor of c-Jun N-terminal kinase (JNK), based on residues 153-163 of JNK-interacting protein-1 (JIP-1). Binds to JNK with affinity…
Product Name: 10Z-HymenialdisineSubtitle: Biological Activity: Biological Activity of 10Z-HymenialdisinePan kinase inhibitor (IC50 values are 6, 10, 22, 28, 35, 40, 70, 80, 100, 470, 500, 600, 700 and 700 nM…
Product Name: SB 706504Subtitle: Biological Activity: Biological Activity of SB 706504p38 MAPK inhibitor. Inhibits LPS-induced transcription of a range of chemokines and cytokines in chronic obstructive pulmonary disease (COPD) monocyte…
Product Name: HG6-64-1Subtitle: Biological Activity: SMLES: N/ACAS NO: 60940-34-3Standard In CHIKey: PAK inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C32H34F3N5O2M.Wt: 577.64General Tips: For obtaining a higher solubility , please warm the…
Product Name: B-Raf IN 1Subtitle: Biological Activity: SMLES: N/ACAS NO: 1025720-94-8Standard In CHIKey: p97 inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C29H24F3N5OM.Wt: 515.53General Tips: For obtaining a higher solubility , please…