Product Name: (3R,4S)-TofacitinibSubtitle: Biological Activity: SMLES: CAS NO: 658084-64-1Standard In CHIKey: Histone_Modification_Research_Compound_Library inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C16H20N6OM.Wt: 312.37General Tips: For obtaining a higher solubility , please warm the…
Product Name: (3S,4R)-TofacitinibSubtitle: Biological Activity: SMLES: CAS NO: 894787-30-5Standard In CHIKey: GPCR/G_protein_Compound_Library inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C16H20N6OM.Wt: 312.37General Tips: For obtaining a higher solubility , please warm the…
Product Name: AZD-9291 mesylateSubtitle: third generation EGFRm inhibitor, oral and irreversibleBiological Activity: SMLES: CAS NO: 6809-52-5Standard In CHIKey: FDA-approved_Drug_Library inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C29H37N7O5SM.Wt: 595.71General Tips: For obtaining…
Product Name: AZD-9291Subtitle: Mutated forms EGFR inhibitorBiological Activity: Biological Activity of AZD-9291Description AZD9291 is a novel oral, potent and selective third generation irreversible inhibitor of mutated forms EGFR with IC50…
Product Name: Mutant EGFR inhibitorSubtitle: Biological Activity: SMLES: C=C/C(O)=N/C1=CC(NC2=NC=C(Cl)C(C3=CNC4=CC=CC=C34)=N2)=C(OC)C=C1N(CCN(C)C)CCAS NO: 228266-40-8Standard In CHIKey: CNS-penetrant_Compound_Library inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C27H30ClN7O2M.Wt: 520.03General Tips: For obtaining a higher solubility , please…
Product Name: (3S,4S)-TofacitinibSubtitle: Biological Activity: SMLES: CAS NO: 1338806-73-7Standard In CHIKey: Clinical_Compound_Library inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C16H20N6OM.Wt: 312.37General Tips: For obtaining a higher solubility , please warm the…
Product Name: AST-1306 TsOHSubtitle: ErbB2 and EGFR inhibitorBiological Activity: Biological Activity of AST-1306 TsOHDescription AST-1306 TsOH is a selective and irreversible inhibitor of ErbB2 and EGFR with IC50 values of…
Product Name: AZD8931 (Sapitinib)Subtitle: ErbB inhibitorBiological Activity: Biological Activity of AZD8931 (Sapitinib)Description AZD8931 is a reversible, ATP competitive inhibitor of EGFR, ErbB2 and ErbB3 with IC50 values of 4 nM,…
Product Name: AST-1306Subtitle: EGFR/HER2 inhibitorBiological Activity: SMLES: CAS NO: 179386-44-8Standard In CHIKey: Apoptosis_Compound_Library inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C24H18ClFN4O2M.Wt: 448.88General Tips: For obtaining a higher solubility , please warm…
Product Name: ARRY-380Subtitle: Tyrosine kinase HER2 and p95-HER2 inhibitorBiological Activity: Biological Activity of ARRY-380Description ARRY-380 is an orally bioavailable, potent, selective, small-molecule inhibitor of tyrosine kinase HER2 and p95-HER2 with…