Product Name: MTEP hydrochlorideSubtitle: MGlu5 antagonistBiological Activity: Biological Activity of MTEP hydrochloridePotent, selective and non-competitive mGlu5 antagonist (IC50 = 5 nM in Ca2+-flux assay; Ki= 16 nM). Displays anxiolytic activity…
Product Name: MPEP HydrochlorideSubtitle: MGlu5 receptor antagonistBiological Activity: Biological Activity of MPEP HydrochloridePotent and highly selective non-competitive antagonist at the mGlu5 receptor subtype (IC50 = 36 nM) and a positive…
Product Name: MK-6892Subtitle: Highly potential GPR109A agonistBiological Activity: SMLES: CC(C)(CC1=NC(=C2C=CC(=O)C=N2)NO1)C(=O)NC3=C(CCCC3)C(=O)OCAS NO: 1234015-52-1Standard In CHIKey: Pyruvate Dehydrogenase inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C19H22N4O5M.Wt: 386.4General Tips: For obtaining a higher solubility…
Product Name: MK-4305Subtitle: OX1/OX2 atagonist,potent and selectiveBiological Activity: Biological Activity of MK-4305Description MK-4305 is a potent antagonist of OX1 receptor and OX2 receptor with Ki values of 0.55 nM and…
Product Name: MK-2894 sodium saltSubtitle: EP4 antagonistBiological Activity: SMLES: CC1=C(C(=C(S1)C)C(=O)NC2(CC2)C3=CC=C(C=C3)C(=O))CC4=CC=C(C=C4)C(F)(F)F.CAS NO: 1403254-99-8Standard In CHIKey: Procollagen C Proteinase inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C25H21F3NNaO3SM.Wt: 495.49General Tips: For obtaining a higher…
Product Name: MK-2894Subtitle: EP4 receptor inhibitorBiological Activity: Biological Activity of MK-2894Description MK-2894 is a highly potent and selective inhibitor of EP4 receptor with IC50 value of 2.5 nM. Targets EP4…
Product Name: MK-0812Subtitle: antagonist of chemokine receptor CCR-2Biological Activity: SMLES: CC(C)C1(CCC(C1)NC2CCOCC2OC)C(=O)N3CCC4=NC=C(C=C4C3)C(F)(F)FCAS NO: 1044870-39-4Standard In CHIKey: Phosphodiesterase PDE) inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C24H34F3N3O3M.Wt: 469.55General Tips: For obtaining a higher…
Product Name: MK 0893Subtitle: Glucagon receptor/IGF-1R antagonistBiological Activity: Biological Activity of MK 0893Description MK 0893 is an inhibitor of both glucagon receptor and IGF-1R with IC50 values of 6.6 nM…
Product Name: mGlu2 agonistSubtitle: Anti-depressants,novel potent agentBiological Activity: SMLES: CC(C(=O)NC1(CC(C2C1C2C(=O)O)SC3=NC=NN3)C(=O)O)N.N.OCAS NO: 1693758-51-8Standard In CHIKey: PDHK inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C13H22N6O6SM.Wt: 390.42General Tips: For obtaining a higher solubility ,…
Product Name: MedetomidineSubtitle: α2-adrenoceptor agonistBiological Activity: SMLES: CC1=C(C(=CC=C1)C(C)C2=CN=CN2)CCAS NO: 1207456-01-6Standard In CHIKey: VPNGEIHDPSLNMU-UHFFFAOYSA-NPAI-1 inhibitorsStandard InChI: InChI=1S/C13H16N2.ClH/c1-9-5-4-6-12(10(9)2)11(3)13-7-14-8-15-13;/h4-8,11H,1-3H3,(H,14,15);1HTyprof Compound: Appearance: Formula: C13H16N2M.Wt: 200.28General Tips: For obtaining a higher solubility , please warm…