Product Name: Plerixafor (AMD3100)Subtitle: CXCR4 chemokine receptor antagonistBiological Activity: SMLES: c1cc(ccc1CN2CCCNCCNCCCNCC2)CN3CCCNCCNCCCNCC3CAS NO: 1446182-94-0Standard In CHIKey: SGLT inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C28H54N8M.Wt: 502.78General Tips: For obtaining a higher solubility…
Product Name: Ki16425Subtitle: LPA receptor antagonistBiological Activity: Biological Activity of Ki16425Antagonist of the lysophosphatidic acid receptors LPA1 and LPA3 (Ki values are 0.25 and 0.36 μM respectively, in a GTPγS…
Product Name: MacitentanSubtitle: Endothelin (ET)(A) and ET(B) receptor antagonistBiological Activity: SMLES: CCCNS(=O)(=O)Nc1c(c(ncn1)OCCOc2ncc(cn2)Br)c3ccc(cc3)BrCAS NO: 760981-83-7Standard In CHIKey: Potassium Channel inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C19H20Br2N6O4SM.Wt: 588.27General Tips: For obtaining a…
Product Name: RamelteonSubtitle: Agonist of melatonin receptor(M1-M2),highly selectiveBiological Activity: Biological Activity of RamelteonDescription Ramelteon is a selective agonist of MT1/MT2 with Ki values of 0.014 nM and 0.045 nM, respectively.…
Product Name: GW9508Subtitle: FFA1/GPR40 agonist,potent and selectiveBiological Activity: Biological Activity of GW9508Potent and selective agonist for the free fatty acid receptor FFA1 (GPR40) (pEC50 values are 7.32, < 4.3 and…
Product Name: CP-945598 HClSubtitle: CB1 antagonist,selective and high affinityBiological Activity: Biological Activity of CP-945598 HClSelective, high affinity CB1 antagonist (Ki values are 0.7 and 0.12 nM in binding and functional…
Product Name: SilodosinSubtitle: α1-adrenoceptor antagonistBiological Activity: Biological Activity of Silodosin 1. Silodosin increases passage of distal ureteral stones. 2. Silodosin temporarily improved LUTS, but did not improve the BOOI after…
Product Name: ScopineSubtitle: Biological Activity: Biological Activity of Scopine 1. Scopine is the metabolite of anisodine, which is a α1-adrenergic receptor agonist . 2. Scopine is a potential brain-targeting moiety…
Product Name: PhloretinSubtitle: A dihydrochalcone found in appleBiological Activity: Biological Activity of Phloretin 1. Phloretin has antimicrobial activity, also against the Gram negative bacteria Salmonella typhimurium ATCC 13311. 2. Phloretin…
Product Name: HydrocortisoneSubtitle: Biological Activity: Biological Activity of Hydrocortisone Adrenal glucocorticoid released in the stress response. Increases glucose production by gluconeogenesis. Immunosuppressant and antidiuretic hormone.SMLES: C12CCC(=O)C=C1CC34CC(O)(C(=O)CO)4(C)C(O)23CAS NO: 1668553-26-1Standard In CHIKey:…