GSK1070916
Product Name: GSK1070916Subtitle: Aurora B/C inhibitorBiological Activity: Biological Activity of GSK1070916Description GSK1070916 is a reversible and ATP-competitive inhibitor of Aurora B and C with IC50 value of 3.5 nM and…
Product Name: GSK1070916Subtitle: Aurora B/C inhibitorBiological Activity: Biological Activity of GSK1070916Description GSK1070916 is a reversible and ATP-competitive inhibitor of Aurora B and C with IC50 value of 3.5 nM and…
Product Name: CYC116Subtitle: Potent Aurora A/B inhibitorBiological Activity: Biological Activity of CYC116Description CYC116 is a potent inhibitor of Aurora A and B with Ki value of 8 nM and 9.2…
Product Name: TAK-901Subtitle: Novel Aurora A/B inhibitorBiological Activity: Biological Activity of TAK-901Description TAK-901 is a novel inhibitor of Aurora A and B with IC50 value of 21 nM and 15…
Product Name: PHA-680632Subtitle: Aurora kinase inhibitor,novel and potentBiological Activity: Biological Activity of PHA-680632Description PHA-680632 is a potent inhibitor of Aurora kinase with IC50 values of 27 nM, 135 nM and…
Product Name: SNS-314 MesylateSubtitle: Aurora A/B/C kinases inhibitor, potent and selectiveBiological Activity: Biological Activity of SNS-314 MesylatePotent, ATP-competitive Aurora kinase inhibitor (IC50 values are 3, 9 and 31 nM for…
Product Name: MK-5108 (VX-689)Subtitle: Aurora-A kinase inhibitor,highly selectiveBiological Activity: Biological Activity of MK-5108 (VX-689)Description MK-5108 is a highly selective inhibitor of Aurora-A kinase with 0.064 nM. Targets Aurora-A IC50 0.064…
Product Name: AMG-900Subtitle: Aurora kinase inhibitorBiological Activity: Biological Activity of AMG-900Description AMG-900 is a potent and highly selective inhibitor of Aurora kinases with IC50 values of 5 nM, 4 nM…
Product Name: HesperadinSubtitle: Aurora B kinase inhibitorBiological Activity: Biological Activity of HesperadinATP-competitive inhibitor of Aurora B kinase (IC50 = 250 nM). Prevents chromosome alignment and segregation; also induces polyploidy and…
Product Name: AT9283Subtitle: Aurora kinase/JAK inhibitorBiological Activity: Biological Activity of AT9283Description AT9283 is a potent inhibitor of Aurora with IC50 values of 3 nM, 3 nM, 1.1 nM, 1.2 nM…
Product Name: JNJ-7706621Subtitle: Potent CDK/Aurora kinase inhibitorBiological Activity: Biological Activity of JNJ-7706621Description JNJ-7706621 is a potent inhibitor of cyclin-dependent kinases (CDK) and Aurora kinases with IC50 values of 9 nM,…