Galanin (2-29) (rat)
Product Name: Galanin (2-29) (rat)Subtitle: Biological Activity: Biological Activity of Galanin (2-29) (rat)Peptide agonist for galanin receptors, showing selectivity for GAL2 (Ki values are 85, 1.9 and 12.6 nM at…
Galanin (1-15) (porcine, rat)
Product Name: Galanin (1-15) (porcine, rat)Subtitle: Biological Activity: Biological Activity of Galanin (1-15) (porcine, rat)N-terminal galanin fragment. In contrast to the full length (1-29) peptide, mediates central cardiovascular effects, perhaps…
BMS 182874 hydrochloride
Product Name: BMS 182874 hydrochlorideSubtitle: ETA antagonistBiological Activity: Biological Activity of BMS 182874 hydrochloridePotent, selective and competitive non-peptide endothelin ETA receptor antagonist (Ki = 48 nM). Displays > 1000-fold selectivity…
BMY 14802 hydrochloride
Product Name: BMY 14802 hydrochlorideSubtitle: Sigma receptor antagonistBiological Activity: Biological Activity of BMY 14802 hydrochloridePotent sigma receptor antagonist (IC50 = 112 nM) with modest to weak affinity for 5-HT1A and…
Ac-RYYRWK-NH2
Product Name: Ac-RYYRWK-NH2Subtitle: Biological Activity: Biological Activity of Ac-RYYRWK-NH2Potent, selective partial agonist peptide for the NOP receptor (Ki = 0.71 nM). Selective over μ, δ and κ opioid receptors (IC50…
[Ala11,22,28]VIP
Product Name: VIPSubtitle: Biological Activity: Biological Activity of VIPPotent and highly selective agonist for the human VPAC1 receptor (Ki values are 7.4 and 2352 nM for binding to human recombinant…
MRS 1334
Product Name: MRS 1334Subtitle: Biological Activity: Biological Activity of MRS 1334Potent and highly selective antagonist for the human adenosine A3 receptor. Ki values are 2.69 nM at hA3, and >…
SB 204070
Product Name: SB 204070Subtitle: Biological Activity: Biological Activity of SB 204070Potent and selective 5-HT4 receptor antagonist (pIC50 = 10.1). Displays >5000-fold selectivity for 5-HT4 over 5-HT1A, 5-HT1D, 5-HT1E, 5-HT2A, 5-HT2C,…
SB 200646 hydrochloride
Product Name: SB 200646 hydrochlorideSubtitle: Biological Activity: Biological Activity of SB 200646 hydrochloride5-HT2C/2B receptor antagonist, selective over 5-HT1A. Affinities are 7.4 (pA2), 6.9 (pKi) and 5.2 (pKi) for 5-HT2B, 2C…
[cPP1-7,NPY19-23,Ala31,Aib32,Gln34] – hPancreatic Polypeptide
Product Name: – hPancreatic PolypeptideSubtitle: Biological Activity: SMLES: N/ACAS NO: 578-74-5Standard In CHIKey: Phospholipase inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C183H281N57O54S2M.Wt: 4207.67General Tips: For obtaining a higher solubility , please…