Product Name: BombesinSubtitle: Biological Activity: Biological Activity of BombesinNeuropeptide with many biological effects including hormone release, stimulation of pancreatic enzyme secretion, inhibition of gastric emptying and modulation of gastric acid…
Product Name: NocIISubtitle: Biological Activity: Biological Activity of NocIIOrphan neuropeptide, flanking nociceptin in the precursor pronociceptin. Stimulates locomotion in mice, possibly through a novel specific receptor.SMLES: N/ACAS NO: 449811-01-2Standard In…
Product Name: Nocistatin (bovine)Subtitle: Biological Activity: Biological Activity of Nocistatin (bovine)An endogenous peptide derived from the same precursor as nociceptin, which is able to block nociceptin-induced allodynia and hyperalgesia and…
Product Name: Nociceptin(1-13)NH2Subtitle: Biological Activity: Biological Activity of Nociceptin(1-13)NH2Potent agonist of the nociceptin (ORL1) receptor, demonstrated both in vitro and in vivo. Selective, competitive antagonism at the nociceptin receptor has…
Product Name: Methysergide maleateSubtitle: Biological Activity: Biological Activity of Methysergide maleateMixed 5-HT1/5-HT2 receptor antagonist.SMLES: O=C(1CN(C)(CC2=CN(C)C3=CC=CC4=C23)C4=C1)N(CO)CC.OC(/C=CC(O)=O)=OCAS NO: 636-00-0Standard In CHIKey: LWYXFDXUMVEZKS-ZVFOLQIPSA-NCathepsin inhibitorsStandard InChI: InChI=1S/C21H27N3O2.C4H4O4/c1-4-15(12-25)22-21(26)14-8-17-16-6-5-7-18-20(16)13(10-23(18)2)9-19(17)24(3)11-14;5-3(6)1-2-4(7)8/h5-8,10,14-15,19,25H,4,9,11-12H2,1-3H3,(H,22,26);1-2H,(H,5,6)(H,7,8)/b;2-1-/t14-,15+,19-;/m1./s1Typrof Compound: Appearance: Formula: C21H27N3O2.C4H4O4M.Wt: 469.54General Tips: For…
Product Name: RS 39604 hydrochlorideSubtitle: Biological Activity: Biological Activity of RS 39604 hydrochlorideA potent and selective 5-HT4 antagonist, with a pKi of 9.1 at 5-HT4 receptors in guinea pig striatal…
Product Name: RS 67333 hydrochlorideSubtitle: Biological Activity: Biological Activity of RS 67333 hydrochlorideA potent and highly selective 5-HT4 partial agonist, with pKi values of 8.7 at 5-HT4 sites in guinea…
Product Name: ICI 215,001 hydrochlorideSubtitle: Biological Activity: Biological Activity of ICI 215,001 hydrochlorideThe active metabolite of ZD 7114.SMLES: N/ACAS NO: 124584-08-3Standard In CHIKey: ATP Citrate Lyase inhibitorsStandard InChI: Typrof Compound:…
Product Name: NociceptinSubtitle: Biological Activity: Biological Activity of NociceptinEndogenous ligand for the NOP opioid receptor (pKi = 8.6). Has no significant activity at μ, δ or κ opioid receptors (pKi…
Product Name: MRS 2179 tetrasodium saltSubtitle: Biological Activity: Biological Activity of MRS 2179 tetrasodium saltA competitive antagonist at P2Y1 receptors (KB = 100 nM). Selective over P2X1 (IC50 = 1.15…