Product Name: m-CPP hydrochlorideSubtitle: Biological Activity: Biological Activity of m-CPP hydrochloride5-HT2C/2B receptor agonist/partial agonist; displays some activity at 5-HT2A and 5-HT1 receptors. pEC50 values are 7.09, 7.2, 6.65, 5.9 and…
Product Name: GR 46611Subtitle: Biological Activity: Biological Activity of GR 466115-HT1D receptor agonist. Blockade of GR 46611-induced hypothermia in the guinea pig provides a useful model with which to study…
Product Name: Pronethalol hydrochlorideSubtitle: Biological Activity: Biological Activity of Pronethalol hydrochlorideβ-adrenergic antagonist, clinically effective in the treatment of angina pectoris and some arrhythmias.SMLES: O(C1=CC=C2C(C=CC=C2)=C1)CNC(C)C.ClCAS NO: 148081-72-5Standard In CHIKey: QONLGXRPRAIDGI-UHFFFAOYSA-NAldehyde Dehydrogenase…
Product Name: SB 203186 hydrochlorideSubtitle: Biological Activity: Biological Activity of SB 203186 hydrochloridePotent 5-HT4 receptor antagonist with high affinity for human atrial 5-HT4 receptors.SMLES: N/ACAS NO: 1797989-42-4Standard In CHIKey: Adenosine…
Product Name: MetaphitSubtitle: Biological Activity: Biological Activity of MetaphitAcylator of PCP and σ-receptors.SMLES: S=C=NC1=CC(C2(CCCCC2)N3CCCCC3)=CC=C1CAS NO: 1782235-14-6Standard In CHIKey: FGSGBQAQSPSRJK-UHFFFAOYSA-NAdenosine Deaminase inhibitorsStandard InChI: InChI=1S/C18H24N2S/c21-15-19-17-9-7-8-16(14-17)18(10-3-1-4-11-18)20-12-5-2-6-13-20/h7-9,14H,1-6,10-13H2Typrof Compound: Appearance: Formula: C18H24N2SM.Wt: 300.46General Tips: For…
Product Name: 2-Methyl-5-hydroxytryptamine hydrochlorideSubtitle: Biological Activity: Biological Activity of 2-Methyl-5-hydroxytryptamine hydrochloride5-HT3 agonist (Ki = 1200 nM) and potent 5-HT6 ligand (Ki = 46 nM).SMLES: CAS NO: 68630-75-1Standard In CHIKey: 5-Lipoxygenase…
Product Name: IPAGSubtitle: Biological Activity: Biological Activity of IPAGPotent σ-receptor antagonist.SMLES: IC1=CC=C(C=C1)N/C(N)=N/23C(C4)C2C4C3CAS NO: 942398-84-7Standard In CHIKey: 5 alpha Reductase inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C17H22IN3M.Wt: 395.29General Tips: For obtaining…
Product Name: L-693,403 maleateSubtitle: Biological Activity: Biological Activity of L-693,403 maleateHigh affinity σ ligand with excellent selectivity over the dopamine D2 receptor.SMLES: N/ACAS NO: 68047-06-3Standard In CHIKey: 15-PGDH inhibitorsStandard InChI:…
Product Name: Octreotide acetateSubtitle: octapeptide congener of native somatostatinBiological Activity: Biological Activity of Octreotide acetatePeptide agonist for sst2, sst3 and sst5 somatostatin receptors. IC50/Kd values (nM) at cloned human somatostatin…
Product Name: Methylprednisolone Sodium SuccinateSubtitle: Biological Activity: SMLES: O1(C(COC(CCC()=O)=O)=O)(C2)(C)(CC1)(C3C)((C)(C=C4)C3=CC4=O)2O.CAS NO: 1642300-78-4Standard In CHIKey: FQISKWAFAHGMGT-SGJOWKDISA-MVDAC inhibitorsStandard InChI: InChI=1S/C26H34O8.Na/c1-14-10-16-17-7-9-26(33,20(29)13-34-22(32)5-4-21(30)31)25(17,3)12-19(28)23(16)24(2)8-6-15(27)11-18(14)24;/h6,8,11,14,16-17,19,23,28,33H,4-5,7,9-10,12-13H2,1-3H3,(H,30,31);/q;+1/p-1/t14-,16-,17-,19-,23+,24-,25-,26-;/m0./s1Typrof Compound: Appearance: Formula: C26H33NaO8M.Wt: 496.53General Tips: For obtaining a higher solubility , please…